Abstract
The Staudinger ligation of phosphine-substituted thioesters with 18F-fluoroethylazide has been successfully applied to access 18F-labelled molecules in radiochemical yields superior to 95%; the first fluorous variant of a Staudinger radio-ligation has been validated.
Original language | English (US) |
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Pages (from-to) | 136-140 |
Number of pages | 5 |
Journal | Organic and Biomolecular Chemistry |
Volume | 9 |
Issue number | 1 |
DOIs | |
State | Published - Jan 1 2011 |
Externally published | Yes |
ASJC Scopus subject areas
- Biochemistry
- Physical and Theoretical Chemistry
- Organic Chemistry