Abstract
As part of continuing studies on drug delivery to the human liver, a phosphonoacetate-trilactoside conjugate (12) has been synthesized in an overall yield of 23%. The shortness of the synthesis of this conjugate hinges upon a successful Michaelis-Arbuzov reaction of bromoacetamide 8 with tris-(trimethylsilyl) phosphite.
Original language | English (US) |
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Pages (from-to) | 335-341 |
Number of pages | 7 |
Journal | Israel Journal of Chemistry |
Volume | 40 |
Issue number | 3-4 |
DOIs | |
State | Published - 2000 |
Externally published | Yes |
ASJC Scopus subject areas
- Chemistry(all)