Synthesis of partially non-peptidic neurotensin mimetics

Dharmpal S. Dood, Alan P. Kozikowski, Bernadette Cusack, Elliott Richelson

Research output: Contribution to journalArticle

Abstract

The synthesis of partially non-peptidic mimetics for NT(8-13) is described. The sequence Arg8Arg9Pro10 of NT(8-13) was replaced by an appropriately substituted indole-2-carboxylate as the non-peptidic equivalent.

Original languageEnglish (US)
Pages (from-to)1241-1246
Number of pages6
JournalBioorganic and Medicinal Chemistry Letters
Volume4
Issue number10
DOIs
StatePublished - May 19 1994
Externally publishedYes

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Neurotensin
neurotensin (9-13)
indole-2-carboxylate

ASJC Scopus subject areas

  • Biochemistry
  • Molecular Biology
  • Organic Chemistry
  • Drug Discovery
  • Pharmaceutical Science

Cite this

Synthesis of partially non-peptidic neurotensin mimetics. / Dood, Dharmpal S.; Kozikowski, Alan P.; Cusack, Bernadette; Richelson, Elliott.

In: Bioorganic and Medicinal Chemistry Letters, Vol. 4, No. 10, 19.05.1994, p. 1241-1246.

Research output: Contribution to journalArticle

Dood, Dharmpal S. ; Kozikowski, Alan P. ; Cusack, Bernadette ; Richelson, Elliott. / Synthesis of partially non-peptidic neurotensin mimetics. In: Bioorganic and Medicinal Chemistry Letters. 1994 ; Vol. 4, No. 10. pp. 1241-1246.
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