Probing Ligand Structure–Activity Relationships in Pregnane X Receptor (PXR): Efavirenz and 8-Hydroxyefavirenz Exhibit Divergence in Activation

Bhargavi Narayanan, Julie M. Lade, Carley J.S. Heck, Kevin D. Dietz, Herschel Wade, Namandjé N. Bumpus

Research output: Contribution to journalArticlepeer-review

2 Scopus citations

Fingerprint

Dive into the research topics of 'Probing Ligand Structure–Activity Relationships in Pregnane X Receptor (PXR): Efavirenz and 8-Hydroxyefavirenz Exhibit Divergence in Activation'. Together they form a unique fingerprint.

Medicine & Life Sciences

Chemical Compounds