Abstract
An expedient synthetic route for 3-aryl β-carbolin-1-ones was developed starting from ethyl acetamidocyanoacetate and chalcone derivatives. The five- and six-membered nitrogen-containing rings in the β-carbolin-1- ones were elaborated efficiently by an intramolecular ketone-nitrile annulation and an intramolecular N-arylation of amide respectively.
Original language | English (US) |
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Pages (from-to) | 1573-1574 |
Number of pages | 2 |
Journal | Organic and Biomolecular Chemistry |
Volume | 2 |
Issue number | 11 |
DOIs | |
State | Published - Jun 7 2004 |
ASJC Scopus subject areas
- Biochemistry
- Physical and Theoretical Chemistry
- Organic Chemistry