Ronnie Mease

Associate Professor

1984 …2020

Research output per year

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Research Output

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Article
2011

High-throughput screen identifies novel inhibitors of cancer biomarker α-methylacyl coenzyme A racemase (AMACR/P504S)

Wilson, B. A. P., Wang, H., Nacev, B. A., Mease, R. C., Liu, J. O., Pomper, M. G. & Isaacs, W. B., May 1 2011, In : Molecular cancer therapeutics. 10, 5, p. 825-838 14 p.

Research output: Contribution to journalArticle

Novel substrate-based inhibitors of human glutamate carboxypeptidase II with enhanced lipophilicity

Plechanovová, A., Byun, Y., Alquicer, G., Škultétyová, LU., Mlčochová, P., Němcová, A., Kim, H. J., Navrátil, M., Mease, R., Lubkowski, J., Pomper, M., Konvalinka, J., Rulíšek, L. & Bařinka, C., Nov 10 2011, In : Journal of medicinal chemistry. 54, 21, p. 7535-7546 12 p.

Research output: Contribution to journalArticle

Strong inhibition of xenografted tumor growth by low-level doses of [32P]ATP

Cheng, Y., Yang, J., Agarwal, R., Green, G. M., Mease, R. C., Pomper, M. G., Meltzer, S. J. & Abraham, J. M., Jun 2011, In : Oncotarget. 2, 6, p. 461-466 6 p.

Research output: Contribution to journalArticle

Open Access
2010

68Ga-labeled inhibitors of prostate-specific membrane antigen (PSMA) for imaging prostate cancer

Banerjee, S. R., Pullambhatla, M., Byun, Y., Nimmagadda, S., Green, G., Fox, J. J., Horti, A., Mease, R. C. & Pomper, M. G., Jul 22 2010, In : Journal of medicinal chemistry. 53, 14, p. 5333-5341 9 p.

Research output: Contribution to journalArticle

Bioisosterism of urea-based GCPII inhibitors: Synthesis and structure-activity relationship studies

Wang, H., Byun, Y., Barinka, C., Pullambhatla, M., Bhang, H. E. C., Fox, J. J., Lubkowski, J., Mease, R. C. & Pomper, M. G., Jan 1 2010, In : Bioorganic and Medicinal Chemistry Letters. 20, 1, p. 392-397 6 p.

Research output: Contribution to journalArticle

Improved syntheses of precursors for PET radioligands [18F]XTRA and [18F]AZAN

Gao, Y., Wang, H., Mease, R. C., Pomper, M. G. & Horti, A. G., Oct 6 2010, In : Tetrahedron Letters. 51, 40, p. 5333-5335 3 p.

Research output: Contribution to journalArticle

Radionuclide based imaging of prostate cancer

Mease, R. C., Oct 22 2010, In : Current topics in medicinal chemistry. 10, 16, p. 1600-1616 17 p.

Research output: Contribution to journalArticle

2009

A low molecular weight PSMA-based fluorescent imaging agent for cancer

Chen, Y., Dhara, S., Banerjee, S. R., Byun, Y., Pullambhatla, M., Mease, R. C. & Pomper, M. G., Dec 18 2009, In : Biochemical and Biophysical Research Communications. 390, 3, p. 624-629 6 p.

Research output: Contribution to journalArticle

Synthesis of [125I]iodoDPA-713: A new probe for imaging inflammation

Wang, H., Pullambhatla, M., Guilarte, T. R., Mease, R. C. & Pomper, M. G., Nov 6 2009, In : Biochemical and Biophysical Research Communications. 389, 1, p. 80-83 4 p.

Research output: Contribution to journalArticle

2008

Interactions between human glutamate carboxypeptidase II and urea-based inhibitors: Structural characterization

Barinka, C., Byun, Y., Dusich, C. L., Banerjee, S. R., Chen, Y., Castanares, M., Kozikowski, A. P., Mease, R. C., Pomper, M. G. & Lubkowski, J., Dec 25 2008, In : Journal of medicinal chemistry. 51, 24, p. 7737-7743 7 p.

Research output: Contribution to journalArticle

N-[N-[(S)-1,3-dicarboxypropyl]carbamoyl]-4-[18F]fluorobenzyl-L- cysteine, [18F]DCFBC: A new Imaging probe for prostate cancer

Mease, R. C., Dusich, C. L., Foss, C. A., Ravert, H. T., Dannals, R. F., Seidel, J., Prideaux, A., Fox, J. J., Sgouros, G., Kozikowski, A. P. & Pomper, M. G., May 15 2008, In : Clinical Cancer Research. 14, 10, p. 3036-3043 8 p.

Research output: Contribution to journalArticle

Radiohalogenated prostate-specific membrane antigen (PSMA)-based ureas as imaging agents for prostate cancer

Chen, Y., Foss, C. A., Byun, Y., Nimmagadda, S., Pullambhatla, M., Fox, J. J., Castanares, M., Lupold, S. E., Babich, J. W., Mease, R. C. & Pomper, M. G., Dec 25 2008, In : Journal of medicinal chemistry. 51, 24, p. 7933-7943 11 p.

Research output: Contribution to journalArticle

Synthesis and evaluation of technetium-99m- and rhenium-labeled inhibitors of the prostate-specific membrane antigen (PSMA)

Banerjee, S. R., Foss, C. A., Castanares, M., Mease, R. C., Byun, Y., Fox, J. J., Hilton, J., Lupold, S. E., Kozikowski, A. P. & Pomper, M. G., Aug 14 2008, In : Journal of medicinal chemistry. 51, 15, p. 4504-4517 14 p.

Research output: Contribution to journalArticle

2005

Radiolabeled small-molecule ligands for prostate-specific membrane antigen: In vivo imaging in experimental models of prostate cancer

Foss, C. A., Mease, R. C., Fan, H., Wang, Y., Ravert, H. T., Dannals, R. F., Olszewski, R. T., Heston, W. D., Kozikowski, A. P. & Pomper, M. G., Jun 1 2005, In : Clinical Cancer Research. 11, 11, p. 4022-4028 7 p.

Research output: Contribution to journalArticle

2004

Preparation of F-18 labeled annexin V: A potential PET radiopharmaceutical for imaging cell death

Toretsky, J., Levenson, A., Weinberg, I. N., Tait, J. F., Üren, A. & Mease, R. C., Aug 1 2004, In : Nuclear Medicine and Biology. 31, 6, p. 747-752 6 p.

Research output: Contribution to journalArticle

2001

Newer methods of labeling diagnostic agents with Tc-99m

Mease, R. C. & Lambert, C., Jan 1 2001, In : Seminars in Nuclear Medicine. 31, 4, p. 278-285 8 p.

Research output: Contribution to journalArticle

Trypanosoma musculi: Tracking parasites and circulating lymphoid cells in host mice

Albright, J. W., Mease, R. C., Lambert, C. & Albright, J. F., Feb 1999, In : Experimental Parasitology. 91, 2, p. 185-195 11 p.

Research output: Contribution to journalArticle

1998

Effects of aging on the dynamics of lymphocyte organ distribution in mice: Use of a radioiodinated cell membrane probe

Albright, J. W., Mease, R. C., Lambert, C. & Albright, J. F., Apr 1 1998, In : Mechanisms of Ageing and Development. 101, 3, p. 197-211 15 p.

Research output: Contribution to journalArticle

1996

Pre-clinical and clinical studies of two new bifunctional chelating agents for immunoscintigraphy with 111in-anti-cea monoclonal antibody

Faivre-Chauvet, A., Chetanneau, A., Bardiès, M., Sai-Maurel, C., Chatal, J. F., Gestin, J. F., Mease, R. C., Meinken, G. E. & Srivastava, S. C., Sep 1996, In : Nuclear medicine communications. 17, 9, p. 781-789 9 p.

Research output: Contribution to journalArticle

Radioiodinated (aminostyryl)pyridinium (ASP) dyes: New cell membrane probes for labeling mixed leukocytes and lymphocytes for diagnostic imaging

Lambert, C., Mease, R. C., Avren, L., Le, T., Sabet, H. & McAfee, J. G., May 1996, In : Nuclear Medicine and Biology. 23, 4, p. 417-427 11 p.

Research output: Contribution to journalArticle

1995

Development and evaluation of copper-67 and samarium-153 labeled conjugates for tumor radioimmunotherapy

Srivastava, S. C., Mausner, L. F., Mease, R. C., Meinken, G. E., Joshi, V., Kolsky, K., Sweet, M. & Steplewski, Z., Jan 1 1995, In : International Journal of Pharmacognosy. 33, SUPPL., p. 92-101 10 p.

Research output: Contribution to journalArticle

Development and evaluation of copper-67 and samarium-153 labeled conjugates for tumor radioimmunotherapy

Srivastava, S. S., Mausner, L. L., Mease, R. R., Meinken, G. G., Joshi, V., Kolsky, K., Sweet, M. & Steplewski, Z., Jan 1 1995, In : Pharmaceutical Biology. 33, S1, p. 92-101 10 p.

Research output: Contribution to journalArticle

1994

Development and evaluation of copper-67 labeled DOTA and TETA immunoconjugates for radioimmunotherapy

Mausner, L. F., Srivastava, S. C., Kolsky, K. L., Mease, R. C., Joshi, V., Meinken, G. E., Kurczak, S., Chatal, J. F. & Steplewski, Z., Jan 1 1994, In : Journal of Labelled Compounds and Radiopharmaceuticals. 35, p. 374-376 3 p.

Research output: Contribution to journalArticle

Production and use of cobalt-55 as an antibody label for PET imaging

Srivastava, S. C., Mausner, L. F., Kolsky, K. L., Mease, R. C., Joshi, V., Meinken, G. E., Pyatt, B., Wolf, A. P., Schlyer, D. J., Levy, A. V. & Fowler, J. S., Jan 1 1994, In : Journal of Labelled Compounds and Radiopharmaceuticals. 35, p. 389-391 3 p.

Research output: Contribution to journalArticle

Reduction in non-specific uptake of indium-111 from using semi-rigid cyclohexyl EDTA immunoconjugates

Srivastava, S. C., Mease, R. C., Meinken, G. E., Gestin, J. F., Joshi, V., Pyatt, B., Mausner, L. F. & Chatal, J. F., Jan 1 1994, In : Journal of Labelled Compounds and Radiopharmaceuticals. 35, p. 303-305 3 p.

Research output: Contribution to journalArticle

1993

Introduction of five potentially metabolizable linking groups between 111In-cyclohexyl EDTA derivatives and F(ab′)2 fragments of anti-carcinoembryonic antigen antibody-I. A new reproducible synthetic method

Gestin, J. F., Faivre-chauvet, A., Mease, R. C., Sai-maurel, C., Thédrez, P., Slinkin, M., Meinken, G. E., Srivastava, S. C. & Chatal, J. F., Aug 1993, In : Nuclear Medicine and Biology. 20, 6, p. 755-762 8 p.

Research output: Contribution to journalArticle

Introduction of five potentially metabolizable linking groups between 111In-cyclohexyl EDTA derivatives and F(ab′)2 fragments of anti-carcinoembryonic antigen antibody-II. Comparative pharmacokinetics and biodistribution in human colorectal carcinoma-bearing nude mice

Faivre-chauvet, A., Gestin, J. F., Mease, R. C., Sai-maurel, C., Thédrez, P., Slinkin, M., Meinken, G. E., Srivastava, S. C. & Chatal, J. F., Aug 1993, In : Nuclear Medicine and Biology. 20, 6, p. 763-771 9 p.

Research output: Contribution to journalArticle

1991

Effect of chelate rigidity on in vivo radioimmunoconjugate distribution

Mease, R. C., Srivastava, S. C., Lambert, C., Meinken, G. E. & Steplewski, Z., Apr 5 1991, In : Journal of Labelled Compounds and Radiopharmaceuticals. 30, p. 319-321 3 p.

Research output: Contribution to journalArticle

Production of no carrier added 80mBr for investigation of Auger electron toxicity

Mease, R. C., DeJesus, O. T., Gatley, S. J., Harper, P. V., Desombre, E. R. & Friedman, A. M., 1991, In : International Journal of Radiation Applications and Instrumentation. Part. 42, 1, p. 57-61 5 p.

Research output: Contribution to journalArticle

Synthesis of new CDTA-linker-antibody systems for improved in-vivo distribution of In-111

Mease, R. C., Gestin, J. F., Meinken, G. E. & Srivastava, S. C., Apr 5 1991, In : Journal of Labelled Compounds and Radiopharmaceuticals. 30, p. 196-197 2 p.

Research output: Contribution to journalArticle

1990

Comparison of the distribution of bromine-77-bromovinyl steroidal and triphenylethylene estrogens in the immature rat

DeSombre, E. R., Hughes, A., Mease, R. C. & Harper, P. V., Jan 1 1990, In : Journal of Nuclear Medicine. 31, 9, p. 1534-1542 9 p.

Research output: Contribution to journalArticle

Development of a new radiolabel (203Pb) and new chelating agents for labeling monoclonal antibodies for imaging.

Srivastava, S. C., Mease, R. C., Meinken, G. E., Mausner, L. F. & Steplewski, Z., 1990, In : Acta radiologica. Supplementum. 374, p. 135-140 6 p.

Research output: Contribution to journalArticle

1988

Bromine-80m-labeled Estrogens: Auger Electron-emitting, Estrogen Receptor-directed Ligands with Potential for Therapy of Estrogen Receptor-positive Cancers

DeSombre, E. R., Mease, R. C., Hughes, A., Harper, P. V., DeJesus, O. T. & Friedman, A. M., Jan 1 1988, In : Cancer Research. 48, 4, p. 899-906 8 p.

Research output: Contribution to journalArticle

Bromine-80m radiotoxicity and the potential for estrogen receptor-directed therapy with auger electrons

DeSombre, E. R., Harper, P. V., Hughes, A., Gatley, S. J., Schwartz, J. L., DeJesus, O. T. & Mease, R. C., Oct 1988, In : Cancer Research. 48, 20, p. 5805-5809 5 p.

Research output: Contribution to journalArticle

Estrogen receptor binding affinity and uterotrophic activity of triphenylhaloethylenes

DeSombre, E. R., Mease, R. C., Sanghavl, J., Singh, T., Seevers, R. H. & Hughes, A., Jun 1988, In : Journal of Steroid Biochemistry. 29, 6, p. 583-590 8 p.

Research output: Contribution to journalArticle

1986

Synthesis and direct estrogen receptor binding affinity of 80mBr-labeled 1,1-bis(p-hydroxyphenyl)-2-bromo-2-phenylethylene

Mease, R. C., DeSombre, E. R. & Hughes, A., Jan 1 1986, In : Journal of Labelled Compounds and Radiopharmaceuticals. 23, 10-12, p. 1397-1399 3 p.

Research output: Contribution to journalArticle

The synthesis of non-steroidal estrogen receptor binding compounds labeled with 80mBr

Seevers, R. H., Mease, R. C., Friedman, A. M. & Desombre, E. R., 1986, In : International Journal of Radiation Applications and Instrumentation.. 13, 4, p. 483-495 13 p.

Research output: Contribution to journalArticle

1984